平安! 发表于 2011-11-9 19:57 p4 D. C- U0 T9 s' ]9 ?' G+ [
Pazopanib (100 mg/kg/day free base equivalent) * u# l& I5 ^3 i4 S
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。/ o, ?0 ]3 [: K
搜索了一下,原料一大堆。
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1 c. @& I2 n4 X& g2 t6 _, W7 [8 u对不起!100mg/kg是用于移植瘤的,我弄错了。
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( W% f' D6 G4 X; u以下是正版说明书的推荐用量。
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o- u( f+ z: F; a) [# W) i--------------------- DOSAGE AND ADMINISTRATION ----------------# \7 U8 t7 C2 [1 Y- M
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1)
! H: W6 M* W. ]( P" K/ z* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
. o7 c$ C* t3 H4 Z# o4 W---------------------DOSAGE FORMS AND STRENGTHS --------------
9 G8 m! C; P3 k200 mg tablets. (3)
3 m: J" q0 c: W; v0 _ q-------------------------------CONTRAINDICATIONS------------------------ |