平安! 发表于 2011-11-9 19:57 ! K1 y2 g# G6 P: Z1 \
Pazopanib (100 mg/kg/day free base equivalent) 1 {& a6 x; A, N4 D/ c' S6 t' ~
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
+ U2 Q, ~# C' r- L搜索了一下,原料一大堆。6 R% s- r- F6 c
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对不起!100mg/kg是用于移植瘤的,我弄错了。
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& h w# e( f8 k T以下是正版说明书的推荐用量。
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--------------------- DOSAGE AND ADMINISTRATION ----------------* S2 d V/ c! p( y
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) - ~+ v0 ]0 ?6 O4 q6 t# j( i# C2 \
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2) : R5 O; g; \9 u" L
---------------------DOSAGE FORMS AND STRENGTHS --------------* G, w& W. S. y2 a& J! K* c( R: Y
200 mg tablets. (3)
5 l. z0 M5 M- k# j, A/ K-------------------------------CONTRAINDICATIONS------------------------ |